(ALPHA-SUBSTITUTED ARALKYLAMINO- AND HETEROARYLALKYLAMINO)PYRIMIDINYL- AND 1,3,5-TRIAZINYLBENZIMIDAZOLES, PHARMACEUTICAL COMPOSITIONS THEREOF AND USE THEREOF IN TREATING PROLIFERATIVE DISEASES Russian patent published in 2017 - IPC C07D403/14 C07D401/04 C07D413/14 C07D401/14 A61K31/53 A61P35/00 

Abstract RU 2608742 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to novel compounds of formula I,

,

having PI3K enzymatic activity.

EFFECT: novel compounds of formula I are obtained, which can be used for regulation of PI3K enzymatic activity, as well as pharmaceutical compositions based thereon.

33 cl, 2 tbl, 63 ex, 3 sch

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RU 2 608 742 C2

Authors

Braun S. Devid

Mettyuz Devid Dzh.

Dates

2017-01-23Published

2012-03-27Filed