NEW AZACYCLIC COMPOUNDS Russian patent published in 2016 - IPC C07D471/10 A61K31/435 A61P3/00 

Abstract RU 2603263 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of formula (I)

,

in which R1 is alkyl, C3-6cycloalkyl, pyrazolyl, phenyl, pyridinyl and the said radicals may contain 1-3 substitutes independently selected from a group comprising alkyl, halogen, haloalkyl, halogenalkoxy group; R2 is phenyl and the said phenyl contains 1-3 substitutes independently selected from a group comprising haloalkyl, halogenalkoxy group; R3 represents hydrogen; A represents -(CH2)n- or -S (O)2-; n equals to 1; or its pharmaceutically acceptable salts.

EFFECT: said compounds can be used as inhibitors of hormone-sensitive lipase.

13 cl, 15 ex

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RU 2 603 263 C2

Authors

Akkermann Zhan

Konte Aurelija

Khuntsiker Daniel

Najdkhart Verner

Nettekofen Mattias

Shults-Gash Tanja

Vertajmer Stenli

Dates

2016-11-27Published

2011-07-08Filed