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(19)

(11)

2 567 395

(13)

(51)

IPC

C07D471/10(2006-01-01)

A61K31/438(2006-01-01)

A61P3/00(2006-01-01)

(21) (22)

Application

2012146875/04, 2011-04-12

(24)

Start date

2011-04-12

(22)

Actual filing date

2011-04-12

(45)

Published

2015-11-10

(72)

Inventor

Akkermann ZhanKonte AurelijaKhuntsiker Daniehl'Najdkhart VernerNettekofen MattiasShul'Ts-Gash Tan'JaVertajmer Stehnli

(73)

Holder

F. Khoffmann-Lja Rosh Ag

AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS Russian patent published in 2015 - IPC C07D471/10 A61K31/438 A61P3/00

Abstract RU 2567395 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds of general formula (I), compositions including the compounds.

EFFECT: compounds for treatment of diabetes, metabolic syndrome and obesity (HSL-inhibitors).

15 cl, 12 ex

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RU 2 567 395 C2

Authors

Akkermann Zhan

Konte Aurelija

Khuntsiker Daniehl'

Najdkhart Verner

Nettekofen Mattias

Shul'Ts-Gash Tan'Ja

Vertajmer Stehnli

Dates

2015-11-10—Published

2011-04-12—Filed