N-PIPERIDIN-3-YL-BENZAMIDE DERIVATIVES FOR CARDIOVASCULAR DISEASES TREATMENT Russian patent published in 2017 - IPC C07D401/14 C07D471/04 C07D487/04 C07D413/14 A61K31/4725 A61K31/4545 A61K31/519 A61P3/06 A61P9/00 

Abstract RU 2618628 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to substituted amide compounds of formula pharmaceutical compositions containing such compounds and application of such compounds for lowering plasma lipid levels, such as low density lipoprotein cholesterol (LDL-cholesterol) and triglycerides, and thus, for treatment of diseases exacerbated by high levels of LDL-cholesterol and triglycerides, such as atherosclerosis and cardiovascular diseases in mammals, including humans.

EFFECT: increased efficiency of compounds application.

42 cl, 10 dwg, 55 ex

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RU 2 618 628 C1

Authors

Darout Etzer

Dullea Robert

Hawkins Julie Jia Li

Londregan Allyn T.

Loria Paula M.

Maguire Bruce

Mcclure Kim F.

Petersen Donna N.

Piotrowski David W.

Dates

2017-05-05Published

2014-04-03Filed