1-IMINO-2,3,4,5-TETRAHYDRO-1H-PYRROLO[3,4-C]PYRIDINE-3,4-DIONES Russian patent published in 2017 - IPC C07D471/04 

Abstract RU 2613967 C1

FIELD: chemistry.

SUBSTANCE: invention relates to methods of obtaining new functionally substituted fused heterocyclic molecules -1-imino-2,3,4,5-tetrahydro-1H-pyrrolo[3,4-c]pyridine-3,4-diones of the formula (I) wherein R1=R2=Me (1a); R1=Me, R2=Et (1b); R1+R2=(CH2)4 (1c); R1+R2=(CH2)5 (1d); R1+R2=(CH2)6 (1e), which may be employed as biologically active compounds in organic synthesis and as fluorescent dyes. The production method consists in suspending the corresponding 2-oxo-4-cyano-1,2-dihydropyridine-3-carboxamide in ethanol, followed by the addition of aqueous ammonia solution with the concentration of 20%, after which the reaction mass is boiled for 30 minutes to obtain the desired product.

EFFECT: new compounds with useful biological activity are obtained.

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RU 2 613 967 C1

Authors

Ershov Oleg Vyacheslavovich

Yatsko Angelina Sergeevna

Fedoseev Sergej Vladimirovich

Ievlev Mikhail Yurevich

Belikov Mikhail Yurevich

Dates

2017-03-22Published

2016-04-25Filed