FIELD: chemistry.
SUBSTANCE: invention relates to a method of producing benzyl ether derivatives of 2-aminonicotinic acid of formula [I] with a high yield and high purity. The method consists in reacting a benzyl halide derivative with a 2-aminonicotinic acid derivative in a polar solvent in the presence of a base.
EFFECT: improved method.
2 cl, 1 tbl, 6 ex
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Authors
Dates
2017-11-15—Published
2013-12-27—Filed