1,6-DIAZABICYCLO[3,2,1]OCTAN-7-ONE DERIVATIVES AND THEIR APPLICATION FOR BACTERIAL INFECTIONS TREATMENT Russian patent published in 2017 - IPC C07D471/08 A61K31/439 A61P31/04 

Abstract RU 2636147 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to application of trans-mono-[2-(N'-[(R)-piperidine-3-carbonyl]hydrazinocarbonyl)-7-oxo-1,6-diazabicyclo[3.2.1]oct-6-yl]ester of sulfuric acid, or a stereoisomer thereof, or a pharmaceutically acceptable salt in combination with cefepime or sulbactam.

EFFECT: prevention or treatment of bacterial infectious disease.

9 cl, 8 tbl, 52 ex

Similar patents RU2636147C1

Title Year Author Number
1,6-DIAZABICYCLO[3,2,1]OCTAN-7-ONE DERIVATIVES AND USING THEM FOR TREATING BACTERIAL INFECTIONS 2012
  • Patel Makhesh Vitkhalbkhaj
  • Deshpande Prasad Keshav
  • Bkhavsar Satish
  • Bkhagvat Sachin
  • Dzhafri Mokhammad Alam
  • Mishra Amit
  • Pavase Laksmikant
  • Gupta Sunil
  • Kale Radzhesh
  • Dzhoshi Sandzhiv
RU2578370C2
PHARMACEUTICAL COMPOSITIONS CONTAINING ANTIBACTERIAL AGENTS 2014
  • Bkhagvat Sakhin
  • Patel Makhesh Vitkhalbkhaj
RU2702361C2
1,6-DIAZABICYCLO[3,2,1]OCTAN-7-ONА DERIVATIVES AND USING THEM IN TREATING BACTERIAL INFECTIONS 2012
  • Bkhagvat Sachin
  • Deshpande Prasad Keshav
  • Bkhavsar Satish
  • Patil Vidzhaikumar Dzhagdishvar
  • Tadipartkhi Ravikumar
  • Pavar Shivadzhi Sampatrao
  • Dzhadkhav Sunil Bkhaginatkh
  • Dabkhade Sandzhaj Kisan
  • Deshmukkh Vikas Vittkhalrao
  • Dond Bkharat
  • Biradzhdar Satish
  • Shaikkh Mokhammad Usman
  • Dekkhane Dipak
  • Patel Pijush Ambalal
RU2570423C2
PHARMACEUTICAL COMPOSITIONS CONTAINING ANTIBACTERIAL AGENTS 2015
  • Patel, Mahesh Vithalbhai
  • Bhagwat, Sachin
  • Satav, Jaykumar Satwaji
  • Khande, Hemant Narendra
  • Joshi, Prashant Ratnakar
  • Palwe, Snehal Rameshwar
RU2705375C2
1,6-DIAZABICYCLO [3,2,1] OCTANE-7-ONA DERIVATIVES AND USE THEREOF FOR TREATING BACTERIAL INFECTIONS 2013
  • Patil Vidzhaikumar Dzhagdishvar
  • Tadipartkhi Ravikumar
  • Dond Bkharat
  • Kale Amol
  • Velupillai Loganatkhan
  • Dekkhane Dipak
  • Biradzhdar Satish Shrimant
  • Shaikkh Mokhammad Usman
  • Maurya Sushilkumar
  • Patel Piyush Ambalal
  • Diksit Prasad
  • Pavar Mangesh
  • Patel Makhesh Vitkhalbkhai
  • Bkhagvat Sachin
RU2614418C2
NITROGEN-CONTAINING BICYCLIC COMPOUNDS 2020
  • Patil, Vijaykumar Jagdishwar
  • Tadiparthi, Ravikumar
  • Bhuniya, Rajib
  • Deshmukh, Vikas Vitthalrao
  • Munshi, Zaki Ahmed Burhanuddin
  • Patel, Piyush Ambalal
  • Joshi, Prashant Ratnakar
  • Chavan, Rajesh
  • Takalkar, Swapna Shripad
  • Yeole, Ravindra Dattatraya
  • Patel, Mahesh Vithalbhai
RU2835672C1
CRYSTALLINE FORMS OF DIAZABICLOCTANE DERIVATIVE AND A METHOD OF THEIR PRODUCTION 2014
  • Abe, Takao
  • Furuuchi, Takeshi
  • Sakamaki, Yoshiaki
  • Mitsuhashi, Nakako
  • Saito, Yumiko
RU2801220C2
CRYSTALLINE FORMS OF DIAZABICYCLOOCTANE DERIVATIVE AND METHOD FOR PRODUCTION THEREOF 2023
  • Abe, Takao
  • Furuuchi, Takeshi
  • Sakamaki, Yoshiaki
  • Mitsuhashi, Nakako
  • Saito, Yumiko
RU2838718C2
CRYSTALLINE FORMS OF DIAZABICYCLOOCTANE DERIVATIVE AND METHOD FOR PRODUCTION THEREOF 2023
  • Abe, Takao
  • Furuuchi, Takeshi
  • Sakamaki, Yoshiaki
  • Mitsuhashi, Nakako
  • Saito, Yumiko
RU2840014C2
CRYSTALLINE FORMS OF DIAZABICYCLOOCTANE DERIVATIVE AND METHOD FOR PRODUCTION THEREOF 2014
  • Abe Takao
  • Furuuti Takesi
  • Sakamaki Josiaki
  • Mitsukhasi Nakako
  • Saito Yumiko
RU2695219C2

RU 2 636 147 C1

Authors

Patel, Makhesh Vitkhalbkhaj

Deshpande, Prasad Keshav

Bkhavsar, Satish

Bkhagvat, Sachin

Dzhafri, Mokhammad Alam

Mishra, Amit

Pavase, Laksmikant

Gupta, Sunil

Kale, Radzhesh

Dzhoshi, Sandzhiv

Dates

2017-11-21Published

2012-08-24Filed