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IPC

C07D487/04(2006-01-01)

A61K31/519(2006-01-01)

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Application

2017121472, 2017-06-19

(24)

Start date

2017-06-19

(22)

Actual filing date

2017-06-19

(45)

Published

2018-01-25

(72)

Inventor

Rasputin Nikolaj AndreevichDemina Nadezhda SergeevnaIrgashev Roman AkhmetovichRusinov Gennadij LeonidovichRusinov Vladimir LeonidovichSpasov Aleksandr AlekseevichBabkov Denis AleksandrovichMajka Olga Yurevna

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Organicheskogo Sinteza Im. I.Ya. Postovskogo Uralskogo Otdeleniya Rossijskoj Akademii Nauk Uro Ran)Federalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Meditsinskij Universitet" Ministerstva Zdravookhraneniya Rossijskoj Federatsii

7-(4-METHOXYPHENYL)-5-PHENYL-4,5-DIHYDRO-[1,2,4]TRIAZOLO[1,5-a]PYRIMIDINE AS ACTIVATOR OF GLUCOKINASE AND INHIBITOR OF DIPEPTIDYL PEPTIDASE OF TYPE 4 AND METHOD OF ITS PRODUCTION Russian patent published in 2018 - IPC C07D487/04 A61K31/519

Abstract RU 2642432 C1

FIELD: chemistry.

SUBSTANCE: invention relates to 7-(4-methoxyphenyl)-5-phenyl-4,5-dihydro-[1,2,4]triazolo [1,5-a]pyrimidine as an activator of glucokinase and an inhibitor of dipeptidyl peptidase of type 4: . The invention also relates to the method of its production.

EFFECT: new compound is produced that can be used as an activator of glucokinase and an inhibitor of dipeptidyl peptidase of type 4.

2 cl, 3 dwg, 3 ex

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RU 2 642 432 C1

Authors

Rasputin Nikolaj Andreevich

Demina Nadezhda Sergeevna

Irgashev Roman Akhmetovich

Rusinov Gennadij Leonidovich

Rusinov Vladimir Leonidovich

Spasov Aleksandr Alekseevich

Babkov Denis Aleksandrovich

Majka Olga Yurevna

Dates

2018-01-25—Published

2017-06-19—Filed