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(19)

(11)

2 644 780

(13)

(51)

IPC

C07C15/20(2006-01-01)

C07D207/10(2006-01-01)

C07D211/22(2006-01-01)

C07D241/04(2006-01-01)

A61K31/40(2006-01-01)

A61K31/435(2006-01-01)

A61K31/495(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2016125777, 2016-06-28

(24)

Start date

2016-06-28

(22)

Actual filing date

2016-06-28

(45)

Published

2018-02-14

(72)

Inventor

Dominique ScholsNadysev Georgij YanovichTikhomirov Aleksandr SergeevichDezhenkova Lyubov GeorgievnaSholts Dominik

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Nauchnoe Uchrezhdenie Institut Po Izyskaniyu Novykh Antibiotikov Imeni G.F. Gauze"

SEMI-SYNTHETIC DERIVATIVES OF HELIOMYCIN INHIBITING TUMOR GROWTH Russian patent published in 2018 - IPC C07C15/20 C07D207/10 C07D211/22 C07D241/04 A61K31/40 A61K31/435 A61K31/495 A61P35/00

Abstract RU 2644780 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to 4-aminomethyl heliomycin derivatives corresponding to the formula:

as well as to pharmaceutical compositions based on them.

EFFECT: technical result: new compounds are obtained with the ability to inhibit the division of tumor cells.

6 cl, 18 ex, 1 tbl

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RU 2 644 780 C2

Authors

Dominique Schols

Nadysev Georgij Yanovich

Tikhomirov Aleksandr Sergeevich

Dezhenkova Lyubov Georgievna

Sholts Dominik

Dates

2018-02-14—Published

2016-06-28—Filed