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(19)

(11)

2 656 853

(13)

(51)

IPC

C07D487/04(2006-01-01)

A61K31/4985(2006-01-01)

A61P25/00(2006-01-01)

A61P35/00(2006-01-01)

A61P37/00(2006-01-01)

(21) (22)

Application

2015107426, 2013-08-19

(24)

Start date

2013-08-19

(22)

Actual filing date

2013-08-19

(45)

Published

2018-06-07

(72)

Inventor

Germann Jokhannes KorneliusKennedi-Smit DzhoshuaLukas Metyu S.Pedilla FernandoShoenfeld Rajan KrejgVovkulich Piter Majkl

(73)

Holder

F. Khoffmann-Lya Rosh Ag

PYRROL[2,3-B]PYRAZINES AS SYK INHIBITORS Russian patent published in 2018 - IPC C07D487/04 A61K31/4985 A61P25/00 A61P35/00 A61P37/00

Abstract RU 2656853 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of the formula .

EFFECT: technical result: new compounds have been obtained, which are the SYK inhibitors and are useful for the treatment of autoimmune and inflammatory diseases.

9 cl, 2 tbl, 38 ex

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RU 2 656 853 C2

Authors

Germann Jokhannes Kornelius

Kennedi-Smit Dzhoshua

Lukas Metyu S.

Pedilla Fernando

Shoenfeld Rajan Krejg

Vovkulich Piter Majkl

Dates

2018-06-07—Published

2013-08-19—Filed