FIELD: chemistry.
SUBSTANCE: invention relates to the novel 4-{2-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-ethyl}-piperidine-1-carboxylic acid methyl amide of formula 1, which has the properties of partial dopamine D2/D3 receptor agonist. 4-{2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl}-piperidine-1-carboxylic acid methylamide corresponds to the formula 1
.
Pharmaceutical composition may, for example, contain from 1 to 2.5 wt% of compound I, from 31 to 31.5 wt% of potato starch and of lactose monohydrate – the rest.
EFFECT: compound may find its application as an active ingredient for a pharmaceutical composition and a drug for treating a psychotic disorder, such as bipolar disorder or certain neurodegenerative diseases.
10 cl, 2 dwg, 7 tbl, 7 ex
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