CRYSTAL FORM α OF COMPOUND OF MONOBENZOATE, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Russian patent published in 2019 - IPC C07D401/04 C07C63/08 C07C51/41 A61K31/53 A61P3/10 

Abstract RU 2677660 C2

FIELD: chemistry.

SUBSTANCE: invention relates to crystalline form α monobenzoate of compound A, a dipeptidyl peptidase-IV inhibitor, of formula (IA). Invention relates also to a method for producing crystalline form α monobenzoate of compound A, to monobenzoate of compound A, to pharmaceutical composition.

(IA).

EFFECT: technical result: obtaining crystalline form α monobenzoate of compound A which is stable and well soluble in water.

9 cl, 2 dwg, 2 tbl, 7 ex

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RU 2 677 660 C2

Authors

Van Vejbo

Li Tunshuan

Tan Sunde

Dates

2019-01-18Published

2015-01-26Filed