BENZOIC ACID, BENZOIC ACID DERIVATIVES AND HETEROARYL CARBOXYLIC ACID CONJUGATES OF OXYCODONE Russian patent published in 2019 - IPC A61K31/485 A61K9/00 A61P25/36 

Abstract RU 2683317 C2

FIELD: chemistry.

SUBSTANCE: group of inventions relates to opioid drugs. Following compounds or their salts are claimed:

, , , .

A composition for use as an opioid agent containing at least one compound or a combination thereof, is also disclosed, and the use of a composition for the manufacture of a drug for a disease treatment, disorder or condition mediated by the binding of at least one opioid to one or more opioid receptors, to reduce or prevent the abuse of drugs or opioids.

EFFECT: group of inventions provides for obtaining new compositions of oxycodone, which have a reduced potential for abuse of oxycodone.

22 cl, 47 dwg, 5 tbl, 4 ex

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RU 2 683 317 C2

Authors

Martin, Andrea K.

Kanski, Jaroslaw

Bera, Bindu

Bera, Sanjib

Guenther, Sven

Mickle, Travis

Dates

2019-03-28Published

2015-11-25Filed