IMIDAZOPYRIDINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY Russian patent published in 2019 - IPC C07D471/04 A61K31/437 A61P3/00 A61P9/00 A61P25/28 A61P27/00 A61P29/00 A61P35/00 A61P37/00

Abstract RU 2683318 C1

FIELD: organic chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to {1-[(2,5-dimethylphenyl)-methyl]imidazo[4,5-b]pyridin-2-yl}(phenyl)methanol. Invention also relates to a pharmaceutical composition based thereon, use thereof and a method of treating and/or preventing rheumatoid arthritis or Crohn's disease.

EFFECT: technical result is obtaining a novel heterocyclic compound useful as a TNFα activity modulator.

4 cl, 1 ex

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RU 2 683 318 C1

Authors

Dzhekson Viktoriya Elizabet

Lekomt Faben Klod

Porter Dzhon Robert

Dates

2019-03-28—Published

2014-12-08—Filed