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(19)

(11)

2 684 644

(13)

(51)

IPC

C07D473/32(2006-01-01)

A61K31/5377(2006-01-01)

A61P1/04(2006-01-01)

A61P19/02(2006-01-01)

(21) (22)

Application

2016127229, 2014-12-08

(24)

Start date

2014-12-08

(22)

Actual filing date

2014-12-08

(45)

Published

2019-04-11

(72)

Inventor

Dzhekson Viktoriya ElizabetKroplin BorisLoue Martin AleksanderPorter Dzhon Robert

(73)

Holder

Ucb Biopharma Sprl

PURINE DERIVATIVES AS TNF ACTIVITY MODULATORS Russian patent published in 2019 - IPC C07D473/32 A61K31/5377 A61P1/04 A61P19/02

Abstract RU 2684644 C1

FIELD: chemical-pharmaceutical industry.

SUBSTANCE: invention relates to a novel purine derivative which is {9-[(2,5-dimethylphenyl)methyl]-2-(morpholin-4-yl)purin-8-yl}methanol.

EFFECT: compound has the properties of a TNF activity modulatorα and can be used for preparing a medicinal agent for treating and/or preventing rheumatoid arthritis or Crohn's disease.

4 cl, 1 ex

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RU 2 684 644 C1

Authors

Dzhekson Viktoriya Elizabet

Kroplin Boris

Loue Martin Aleksander

Porter Dzhon Robert

Dates

2019-04-11—Published

2014-12-08—Filed