SUBSTITUTED 1,2,5-TRIMETHYL- AND 2,2,6,6-TETRAMETHYL-4-AMINOPIPERIDINES, HAVING ANTI-ISCHEMIC ACTIVITY Russian patent published in 2019 - IPC C07D211/66 C07D401/12 A61K31/44 A61K31/4468 A61P9/10 

Abstract RU 2686317 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a new group of substituted polyalkyl-4-aminopiperidines of general formula (Ia, b) 1a 1b and pharmaceutically acceptable salts thereof, preferably hydrochlorides of general formula (Ia, b ⋅ HCl). Disclosed compounds have cardiotropic, particularly anti-ischemic activity.

EFFECT: substituted 1,2,5-trimethyl- and 2,2,6,6-tetramethyl-4-aminopiperidines possessing anti-ischemic activity are proposed.

5 cl, 1 dwg, 2 tbl, 6 ex

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RU 2 686 317 C2

Authors

Seredenin Sergej Borisovich

Kostochka Leonid Mikhajlovich

Kryzhanovskij Sergej Aleksandrovich

Tsorin Iosif Borisovich

Vititnova Marina Borisovna

Stolyaruk Valerij Nikolaevich

Gudasheva Tatyana Aleksandrovna

Dates

2019-04-25Published

2015-04-24Filed