PHARMACEUTICAL COMPOSITION BASED ON N-BENZYL-N-METHYL-1-PHENYLPYRROLO [1,2-A] PYRAZINE-3-CARBOXAMIDE Russian patent published in 2019 - IPC A61K31/4985 A61K9/20 A61K9/48 A61K47/38 A61K47/58 A61K47/04 A61K47/10 A61P25/22 

Abstract RU 2689396 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to a pharmaceutical composition having anxiolytic activity. Pharmaceutical composition for preparing a solid dosage form contains N-benzyl-N-methyl-1-phenylpyrrolo[1,2-a]pyrazine-3-carboxamide and pharmaceutically acceptable excipients in said ratio, wt. %: N-benzyl-N-methyl-1-phenylpyrrolo[1,2-a]pyrazine-3-carboxamide - 1.0; microcrystalline cellulose - 88.0; cross-linked polyvinylpyrrolidone - 4.0; polyvinylpyrrolidone - 6.0; magnesium stearate 1.0.

EFFECT: invention provides extending the range of medications possessing anxiolytic action, increases bioavailability of the active substance due to the excipients used.

3 cl, 7 tbl, 7 ex

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RU 2 689 396 C2

Authors

Seredenin Sergej Borisovich

Gudasheva Tatyana Aleksandrovna

Alekseev Konstantin Viktorovich

Blynskaya Evgeniya Viktorovna

Yudina Darya Valentinovna

Mikheeva Anna Sergeevna

Durnev Andrej Dmitrievich

Mokrov Grigorij Vladimirovich

Yarkova Milada Alnordovna

Zherdev Vladimir Pavlovich

Kolyvanov Gennadij Borisovich

Litvin Aleksandr Alekseevich

Dates

2019-05-28Published

2017-07-06Filed