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2 734 240

(13)

C2

(51)

IPC

C07D487/04(2006-01-01)

A61K31/4985(2006-01-01)

A61P25/00(2006-01-01)

(21) (22)

Application

2018140021, 2018-11-13

(24)

Start date

2018-11-13

(22)

Actual filing date

2018-11-13

(45)

Published

2020-10-13

(72)

Inventor

Seredenin Sergej BorisovichMokrov Grigorij VladimirovichYarkova Milada AlnordovnaPantileev Andrej SergeevichGudasheva Tatyana AleksandrovnaDurnev Andrej Dmitrievich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Nauchnoe Uchrezhdenie Institut Farmakologii Imeni V.V. Zakusova"

DIPHENYLPYRROLO[1,2-A]PYRAZINE-3-CARBOXAMIDES-COMPOUNDS HAVING NEUROPSYCHOTROPIC ACTIVITY, METHODS FOR PREPARING THEM Russian patent published in 2020 - IPC C07D487/04 A61K31/4985 A61P25/00 

Abstract RU 2734240 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to 1-phenyl-N-phenylpyrrolo[1,2-a]pyrazine-3-carboxamides of general formula (1):

,

where R can be hydrogen, (C1-C4)-alkyl or benzyl group, as well as their method of producing and method of treating disorders, mediated by their activity.

EFFECT: technical result is obtaining novel compounds having anxiolytic activity.

7 cl, 5 tbl, 5 ex

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RU 2 734 240 C2

Authors

Seredenin Sergej Borisovich

Mokrov Grigorij Vladimirovich

Yarkova Milada Alnordovna

Pantileev Andrej Sergeevich

Gudasheva Tatyana Aleksandrovna

Durnev Andrej Dmitrievich

Dates

2020-10-13—Published

2018-11-13—Filed

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