1,3,4-OXADIAZOLE SULPHAMIDE DERIVATIVES AS HISTONE DEACETYLASE 6 INHIBITOR AND PHARMACEUTICAL COMPOSITION CONTAINING THEM Russian patent published in 2019 - IPC C07D271/10 C07D413/12 A61K31/4245 A61P3/00 A61P1/00 A61P9/00 A61P17/00 A61P19/00 A61P25/00 

Abstract RU 2695227 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds of formula I, stereoisomers thereof or pharmaceutically acceptable salts thereof, as well as pharmaceutical compositions based thereon and a method of treating mediated diseases.

[Formula I]

EFFECT: obtaining novel compounds having histone deacetylase inhibitory activity.

10 cl, 2 tbl, 78 ex

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RU 2 695 227 C1

Authors

Lee, Jaekwang

Han, Younghue

Kim, Yuntae

Min, Jaeki

Bae, Miseon

Kim, Dohoon

Jin, Seokmin

Kyung, Jangbeen

Dates

2019-07-22Published

2016-07-27Filed