METHOD OF PRODUCING PYRIMIDINYLCYCLOPENTANE COMPOUNDS Russian patent published in 2019 - IPC C07D239/70 C07C269/06 C07C271/22 

Abstract RU 2702355 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing a compound of formula (I)

comprising a reaction of coupling a compound of formula

with a compound of formula (III),

where M is Na+.

EFFECT: technical result is a novel method of producing a compound of formula (I), which increases stereoselectivity, simplifies purification, reduces the number of reaction steps, improves overall yield, increases efficiency, environmental purity and cost.

66 cl, 5 tbl, 16 ex

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Authors

Iding Khans

Reents Rajnkhard

Skalone Mikelandzhelo

Gosselen Fransis

Dates

2019-10-08Published

2014-11-13Filed