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2 724 334

(13)

(51)

IPC

C07D209/42(2006-01-01)

C07D401/12(2006-01-01)

C07D403/12(2006-01-01)

C07D413/12(2006-01-01)

A61K31/404(2006-01-01)

A61K31/04(2006-01-01)

A61K31/06(2006-01-01)

A61P31/06(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2019113030, 2016-11-10

(24)

Start date

2016-11-10

(22)

Actual filing date

2016-11-10

(45)

Published

2020-06-23

(72)

Inventor

Apt Aleksandr SolomonovichVelezheva Valeriya SergeevnaNikonenko Boris VladimirovichKornienko Albert GrigorevichMajorov Konstantin BorisovichIvanov Pavel YurevichKondrateva Tatyana KonstantinovnaKorotetskaya Marina ValerevnaSalina Elena Gennadevna

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Elementoorganicheskikh Soedinenij Im. A.N.Nesmeyanova Rossijskoj Akademii Nauk Ran)

3-TRIAZENONE INDOLES POSSESSING MYCOBACTERIUM ACTIVITY Russian patent published in 2020 - IPC C07D209/42 C07D401/12 C07D403/12 C07D413/12 A61K31/404 A61K31/04 A61K31/06 A61P31/06 A61P31/04

Abstract RU 2724334 C1

FIELD: chemistry.

SUBSTANCE: invention refers to compounds having antimycobacterial activity. More specifically, it relates to substituted 3-triazenone indoles, having activity against various mycobacteria, including against their multidrug-resistant strains.

EFFECT: substituted 3-triazenone indoles showed high in vitro activity against isoniazid-resistant strain M_ tuberculosis and M_avium.

4 cl, 1 dwg, 2 tbl, 10 ex

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RU 2 724 334 C1

Authors

Apt Aleksandr Solomonovich

Velezheva Valeriya Sergeevna

Nikonenko Boris Vladimirovich

Kornienko Albert Grigorevich

Majorov Konstantin Borisovich

Ivanov Pavel Yurevich

Kondrateva Tatyana Konstantinovna

Korotetskaya Marina Valerevna

Salina Elena Gennadevna

Dates

2020-06-23—Published

2016-11-10—Filed