HYDROCHLORIDES OF SUBSTITUTED 2-[(DIMETHYLAMINO)METHYL]ARYLDIMETHYL CARBAMATES EXHIBITING ANTICHOLINESTERASE ACTIVITY Russian patent published in 2021 - IPC C07C271/44 A61K31/27 A61K31/325 A61P39/02 

Abstract RU 2754133 C1

FIELD: medicine.

SUBSTANCE: invention relates to the field of medicine, namely to an application of centrally active hydrochlorides of substituted 2-[(dimethylamino)methyl]aryldimethyl carbamates by the general formula I as reversible inhibitors of acetyl cholinesterase, potentially applicable in treating poisonings from antidepressants, organophosphorous and cholinotropic compounds. Invention also relates to new hydrochlorides of 2-[(dimethylamino)methyl]aryldimethyl carbamates.

EFFECT: technical result is a new application of hydrochlorides of substituted 2-[(dimethylamino)methyl]aryldimethyl carbamates for treating poisonings.

2 cl, 2 tbl, 5 ex

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RU 2 754 133 C1

Authors

Bespalov Aleksandr Yakovlevich

Prokopenko Lyubov Ivanovna

Gorchakova Tatyana Leonidovna

Kozlov Viktor Konstantinovich

Petrov Aleksandr Nikolaevich

Zajtseva Mariya Anatolevna

Melekhova Aleksandra Sergeevna

Belskaya Alisa Vladimirovna

Melnikova Margarita Viktorovna

Ivanov Maksim Borisovich

Chigareva Svetlana Mikhajlovna

Dates

2021-08-27Published

2020-08-04Filed