FIELD: pharmaceuticals.
SUBSTANCE: invention relates to compounds of formula I, where the values A, B, C, L, R2, R3, R7-R9, m, p are specified in the claims, which are selective allosteric inhibitors of EGFR mutant variants containing T790M/L858R, T790M/L858R/C797S, L858R, L858R/C797S and to pharmaceutical compositions containing these compounds.
EFFECT: compounds can be used in the preparation of an agent for the therapeutic and/or prophylactic treatment of non-small cell lung cancer characterized by mutations activating EGFR.
15 cl, 8 tbl, 68 ex
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