TRIAZOLE DERIVATIVE, METHOD FOR PRODUCTION THEREOF AND USE THEREOF Russian patent published in 2024 - IPC C07D403/06 A61K31/506 A61P27/02 A61P31/12 A61P35/00 A61P37/08 

Abstract RU 2832307 C2

FIELD: pharmaceutics.

SUBSTANCE: invention refers to pharmaceutics, namely to a triazole derivative of formula I. Invention also relates to a pharmaceutical composition based on the compound of formula I and use of the compound of formula I for preparing a drug for treating a disorder associated with CRM1 activity. I.

EFFECT: obtaining a compound of formula I having CRM1 inhibitory activity for treating CRM1-mediated diseases.

6 cl, 1 dwg, 3 tbl, 1 ex

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RU 2 832 307 C2

Authors

Zhu, Yongqiang

Lei, Meng

Miao, Hang

Wang, Xueyuan

Dates

2024-12-23Published

2022-03-11Filed