METHOD OF PREPARING ENANTIOMERICALLY PURE AZETIDINE-2-CARBOXYLIC ACID Russian patent published in 2001 - IPC

Abstract RU 2163595 C2

FIELD: chemical industry. SUBSTANCE: described is method of preparing enantiomerically pure azetidine-2-carboxylic acid (AzeOH) by dissolving racemic mixture AzeOH and L or D-tartaric acid in solvents to form homogeneous solution, selective crystallization of the resulting pure AzeOH tartrate from solution followed by isolation of pure amino acid. Also described are new L-azetidine-2-carboxylic acid D-tartrate and D-azetidine-2-carboxylic acid L-tartrate. EFFECT: product with higher yield and greater optical purity by method using less stages. 16 cl, 11 ex

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Authors

Bart Filipp

Frichi Khugo

Njustrem Jan-Ehrik

Pfenninger Armin

Dates

2001-02-27Published

1996-06-24Filed