FIELD: organic chemistry, medicine, pharmacy.
SUBSTANCE: invention relates to new derivatives of artemisinin of the general formula (I):
wherein Y has values given in the description, and also to a method for their preparing, pharmaceutical compositions containing these C-10-substituted derivatives, and to a method for treatment of infectious diseases caused by parasite. Invention provides preparing new compounds that can be used for treatment of malaria, neosporosis and coccidiosis.
EFFECT: improved preparing method, valuable medicinal properties of compounds.
19 cl, 9 tbl, 62 ex
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Authors
Dates
2004-09-20—Published
1999-07-14—Filed