FIELD: organic chemistry, medicine.
SUBSTANCE: invention relates to new derivative of phenylpiperazine mesylate of the formula: 
possessing preferable properties as compared with form of a free base of the same compound. Also, invention describes a pharmaceutical composition and a method for inhibition of activity of dopamine D2-receptors and site of serotonin reuptake.
EFFECT: valuable pharmacological properties of derivatives.
3 cl, 1 ex
| Title |
Year |
Author |
Number |
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2002 |
- Fenstra Rulof V.
- Ronken Ehrik
- Krjuse Kornelis G.
- Makkriri Ehndrju S.
- Van Skharrenburg Gustaf J.M.
|
RU2279431C2 |
| ORGANIC COMPOUNDS |
2017 |
|
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2012 |
|
RU2613177C2 |
| PYRIDINE DERIVATIVES USED AS QUICKLY DISSOCIABLE DOPAMINE RECEPTOR 2 ANTAGONISTS |
2008 |
- Makdonal'D Gregor Dzhejms
- Bartolome-Nebreda Khose Manuehl'
- Van Gol Mikhil' Ljuk Marija
- Del'Gado-Khimenes Fransiska
|
RU2480462C2 |
| NEW PHENYLPIPERAZINES |
2000 |
- Van Khes Rulof
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- Krjuse Kornelis G.
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|
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1995 |
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- Klotet Khoan Uget
- Fransisko Markil'Jas Olondris
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- Anna Bosh Rovira
- Khoan Roka Asin
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|
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2018 |
- Ivashchenko Aleksandr Vasilevich
- Nikitin Aleksandr Vladimirovich
- Karapetyan Ruben Navasardovich
- Kuznetsova Anastasiya Aleksandrovna
|
RU2677268C1 |
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2004 |
- Langen Barbara
- Rundfel'Dt Kris
- Dost Rita
- Ljuddens Khartmut
- Rabe Khol'Ger
|
RU2354377C2 |
| 4-ALKOXYPYRIDAZINE DERIVATIVES AS FAST DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS |
2008 |
- Makdonal'D Gregor Dzhejms
- Bartolome-Nebreda Khose Manuehl'
|
RU2464268C2 |
| LIGAND WITH WIDE RANGE OF SIMULTANEOUS RECEPTOR ACTIVITY, PHARMACEUTICAL COMPOSITION, METHOD OF PREPARING SAID COMPOSITION AND MEDICINAL AGENT |
2008 |
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|
RU2374245C1 |
