FIELD: chemistry.
SUBSTANCE: invention relates to 5'-phosphorus-containing derivatives of 2',3'-dideoxy-3'-thiacytidine with general structural formula given below 
, where R=H, NH2-C(O)-. The invented compounds can be used for inhibiting reproduction of the human immunodeficiency virus type 1 in an MT-4 cell culture.
EFFECT: increased antiviral activity of the compounds.
1 cl, 2 tbl, 4 ex
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