METHOD OF PRODUCING INDOLIZINO[7,6-b]INDOLE DERIVATIVES Russian patent published in 2012 - IPC C07D487/12 

Abstract RU 2439073 C1

FIELD: chemistry.

SUBSTANCE: present invention relates to organic chemistry and specifically to a method of producing indolizino[7,6-b]indole derivatives of formulae Ia-f , where Ia: R=R1=R2=H; Ib: R-R2=H, R1=CH3; Ic: R=H, R1=CH3, R2=Cl; Id: R=Cl, R1=R2=H; Ie: R=CH3, R1=H, R2=Cl; If: R=OCH3, R1=H, R2=Cl, which involves reaction of 3-alkyl-5-tosyl-5H-pyrido[4,3-b]indole II and phenacyl bromide in a mixture of benzene and toluene.

EFFECT: novel heterocyclic backbone - indolizino[7,6-b]indole derivatives.

1 cl, 2 tbl, 2 ex

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RU 2 439 073 C1

Authors

Pilipenko Arkadij Sergeevich

Uchuskin Maksim Grigor'Evich

Butin Aleksandr Valerianovich

Trushkov Igor' Vladimirovich

Dates

2012-01-10Published

2010-07-13Filed