7-MEMBER CYCLIC COMPOUNDS, SYNTHESIS METHODS THEREOF AND PHARMACEUTICAL APPLICATION THEREOF Russian patent published in 2012 - IPC C07D243/08 C07D401/06 C07D405/06 C07D405/12 C07D409/12 C07D413/12 A61K31/551 A61P9/00 A61P5/28 

Abstract RU 2448099 C2

FIELD: chemistry.

SUBSTANCE: described are novel 7-member heterocyclic compounds of general formula (values of radicals are given in the claim) or salts thereof or solvates thereof having chymase inhibiting activity and suitable for preventing or treating different diseases in which chymase is involved, a method of producing said compounds, intermediate compounds and a pharmaceutical composition for preventing or treating diseases in which chymase is involved, including compounds of formula (I) or pharmaceutically acceptable salts or solvates thereof.

EFFECT: improved properties of the compound.

23 cl, 12 tbl, 308 ex

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RU 2 448 099 C2

Authors

Muto Tsuesi

Tanaka Taisaku

Maruoka Khirosi

Imadzo Seiiti

Tomimori Esiaki

Dates

2012-04-20Published

2005-12-01Filed