N-OXIDE AND/OR DI-N-OXIDE DERIVATIVES OF STABILISERS/MODULATORS OF DOPAMINE RECEPTORS, DEMONSTRATING IMPROVED PROFILES OF CARDIO-VASCULAR SIDE EFFECTS Russian patent published in 2012 - IPC C07D211/94 A61K31/451 A61P25/00 

Abstract RU 2470013 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to N-oxide and/or di-N-oxide derivatives of stabilisers/modulators of dopamine receptors, which have formula (2) (given in description) and to their pharmaceutical preparations, containing said compounds.

EFFECT: invention relates to application of said compounds for treating central nervous system disorders, in particular, for treatment of dopamine-mediated disorders, such as motor disorders, psychoses, anxiety disorders, impaired development of nerves, sleep disorders and disorders, associated with substances.

9 cl, 2 dwg

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RU 2 470 013 C2

Authors

Vikstrem Khokan V.

Dates

2012-12-20Published

2008-04-11Filed