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(19)

(11)

2 471 786

(13)

(51)

IPC

C07D243/14(2006-01-01)

C07D239/50(2006-01-01)

A61K31/505(2006-01-01)

A61K31/5513(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2011134966/04, 2011-08-19

(24)

Start date

2011-08-19

(22)

Actual filing date

2011-08-19

(45)

Published

2013-01-10

(72)

Inventor

Egorova Alevtina Jur'EvnaTerentjuk Georgij SergeevichGrinev Vjacheslav Sergeevich

(73)

Holder

Federal'Noe Gosudarstvennoe Bjudzhetnoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet Imeni N.G. Chernyshevskogo"

AGENT FOR CANCER THERAPY Russian patent published in 2013 - IPC C07D243/14 C07D239/50 A61K31/505 A61K31/5513 A61P35/00

Abstract RU 2471786 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to new compounds described by general formulas specified below, in the free form as pharmaceutically acceptable salts possessing anticancer activity and may be applicable in medical practice as a therapeutic agent for treating cancer. The compounds under the present invention are described by one of structure formulas: or wherein Ar represents Ph or 4-NO₂-C₆H₄.

EFFECT: presented compounds enable reducing or eliminating completely tumour cell growth by disturbing cell division at the level of enzyme inhibition.

1 tbl, 5 ex

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RU 2 471 786 C1

Authors

Egorova Alevtina Jur'Evna

Terentjuk Georgij Sergeevich

Grinev Vjacheslav Sergeevich

Dates

2013-01-10—Published

2011-08-19—Filed