ETHYL 5-ALKYL-7,7-DIMETHYL-2',9,11-TRIOXO-5'-PHENYL-1',2',5,6,7,8,9,11-OCTAHYDROSPIRO{INDENO[1,2-b][QUIOLINE-10,3'-PYRROL}-4'-CARBOXYLATES AND METHOD FOR PREPARING THEM Russian patent published in 2013 - IPC C07D471/10 

Abstract RU 2485120 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to organic chemistry, namely to new individual compounds of spiro{indeno[1,2-b]quinoline-10,3'-pyrroles}, namely to ethyl 5-alkyl-7,7-dimethyl-2',9,11-trioxo-5'-phenyl- 1',2', 5,6,7,8,9,11-octahydrospiro{indeno[1,2-6]quinoline-10,3'-pyrrol}-4'-carboxylates of general formula wherein R=CH2Ph, C6H11-c, Ph, C6H4OMe-4, C6H4Me-4; Alk=CH2Ph, All; furthermore, the invention refers to a method for preparing them.

EFFECT: preparing the new compounds which may be used as initial products for synthesis of new heterocyclic systems and in pharmacology as those exhibiting analgesic activity.

4 cl, 1 tbl

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RU 2 485 120 C1

Authors

Dmitriev Maksim Viktorovich

Silajchev Pavel Sergeevich

Makhmudov Ramiz Ragibovich

Maslivets Andrej Nikolaevich

Dates

2013-06-20Published

2012-02-07Filed