Show metadata Hide metadata

(19)

(11)

2 502 733

(13)

(51)

IPC

C07D209/30(2006-01-01)

C07D401/06(2006-01-01)

C07D409/08(2006-01-01)

A61K31/404(2006-01-01)

A61P25/04(2006-01-01)

(21) (22)

Application

2010143451/04, 2009-03-25

(24)

Start date

2009-03-25

(22)

Actual filing date

2009-03-25

(45)

Published

2013-12-27

(72)

Inventor

Tsemol'Ka ZaskijaShunk ShtefanNol'Te BertLints KlausShreder Vol'FgangEhngl'Berger VernerShik KhansZonnenshajn KhajmutKhenkel' BirgittaBalint Jozhev

(73)

Holder

Grjunental' Gmbkh

ARYLCYCLOHEXANE DERIVATIVES Russian patent published in 2013 - IPC C07D209/30 C07D401/06 C07D409/08 A61K31/404 A61P25/04

Abstract RU 2502733 C2

FIELD: chemistry.

SUBSTANCE: invention relates to (hetero)arylcyclohexane derivatives of formula , where values of Y₁, Y₁', Y₂, Y₂', Y₃, Y₃', Y₄, Y₄', R₁-R₃ are given in the first claim, having affinity for the µ- opioid receptor and ORL 1-receptor.

EFFECT: enabling use of the derivatives in drugs for treating pain.

10 cl, 2 tbl, 40 ex

Similar patents RU2502733C2

Title	Year	Author	Number
SPIRO(5,5)UNDECANE DERIVATIVES	2009	Zaskia Tsemol'Ka Shtefan Shunk Klaus Lints Vol'Fgang Shreber Verner Ehngl'Berger Fritts Tajl' Birgit Roloff	RU2515895C2
SUBSTITUTED DERIVATIVES OF 4-AMINOCYCLOHEXANE	2009	Bert Nol'Te Vol'Fgang Shreder Klaus Lints Verner Ehngl'Berger Khans Shik Khajnts Graunbaum Birgit Roloff Zigrid Otsegovski Jozhev Balint Khel'Mut Zonnenshajn	RU2532545C2
SUBSTITUTED DERIVATIVES OF 4-AMINOCYCLOHEXANE	2009	Bert Nol'Te Vol'Fgang Shreder Klaus Lints Verner Ehngl'Berger Khans Shik Khajnts Graubaum Birgit Roloff Zigrid Otsegovski Jozhev Balint Khel'Mut Zonnenshajn	RU2525236C2
SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES	2009	Nol'Te Bert Shreder Vol'Fgang Lints Klaus Ehngl'Berger Verner Shik Khans Graubaum Khajnts Roloff Birgit Otsegovki Zigrid Balint Jozhev Zonnenshajn Khel'Mut	RU2503660C2
SUBSTITUTED CYCLOHEXYLDIAMINES	2009	Zaskija Tsemol'Ka Bert Nol'Te Klaus Lints Derek Dzhon Sonders Vol'Fgang Shreder Verner Ehngl'Berger Fritts Tajl' Khans Shikk Jens Kaufmann Julian Gebauer Khel'Mut Zonnenshajn	RU2526251C2
HYDROXYMETHYL CYCLOHEXYLAMINES	2009	Sven Frormann Zaskija Tsemol'Ka Klaus Lints Verner Ehngl'Berger Fritts Tajl'	RU2514192C2
DERIVATIVES OF SUBSTITUTED SPIROCYCLIC CYCLOHEXANE	2009	Tsemol'Ka Zaskija Nol'Te Bert Frormann Sven Khintse Klaudia Lints Klaus Shreder Vol'Fgang Ehngl'Berger Verner Shik Khans Zonnenshajn Khel'Mut	RU2497824C2
SUBSTITUTED HETEROARYL DERIVATIVES	2007	Tsemol'Ka Zaskja Shunk Shtefan Ehngl'Berger Verner Kegel' Babette-Ivonne Lints Klaus Shik Khans Zonnenshajn Khel'Mut Graubaum Khajnts Khintse Klaudia	RU2459806C2
SUBSTITUTED PHENYLUREAS AND PHENYLAMIDES AS LIGANDS OF VANILLOID RECEPTORS	2010	Robert Frank Gregor Barenberg Tomas Kristof Klaus Shine Zhan De-Vri Nil'S Damann Sven Frormann Bernkhard Lesh Chzhiu Li Ensu Kim Mensop Kim	RU2553392C2
SUBSTITUTED 2-OXO- AND 2- THIOXO- DIHYDROQUINOLINE-3-CARBOXAMIDES AS KCNQ2/3 MODULATORS	2011	Kjunert Sven Barenberg Gregor Kless Akhim Shreder Volfgang	RU2581362C2

RU 2 502 733 C2

Authors

Tsemol'Ka Zaskija

Shunk Shtefan

Nol'Te Bert

Lints Klaus

Shreder Vol'Fgang

Ehngl'Berger Verner

Shik Khans

Zonnenshajn Khajmut

Khenkel' Birgitta

Balint Jozhev

Dates

2013-12-27—Published

2009-03-25—Filed