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(19)

(11)

2 459 806

(13)

(51)

IPC

C07D209/08(2006-01-01)

C07D209/14(2006-01-01)

C07D209/12(2006-01-01)

C07D209/20(2006-01-01)

C07D401/06(2006-01-01)

C07D403/06(2006-01-01)

C07D409/08(2006-01-01)

C07D413/06(2006-01-01)

C07D417/06(2006-01-01)

C07D471/04(2006-01-01)

C07D307/81(2006-01-01)

A61K31/404(2006-01-01)

A61K31/4178(2006-01-01)

A61P25/00(2006-01-01)

A61P9/00(2006-01-01)

A61P1/00(2006-01-01)

(21) (22)

Application

2009105398/04, 2007-07-17

(24)

Start date

2007-07-17

(22)

Actual filing date

2007-07-17

(45)

Published

2012-08-27

(72)

Inventor

Tsemol'Ka ZaskjaShunk ShtefanEhngl'Berger VernerKegel' Babette-IvonneLints KlausShik KhansZonnenshajn Khel'MutGraubaum KhajntsKhintse Klaudia

(73)

Holder

Grjunental' Gmbkh

SUBSTITUTED HETEROARYL DERIVATIVES Russian patent published in 2012 - IPC C07D209/08 C07D209/14 C07D209/12 C07D209/20 C07D401/06 C07D403/06 C07D409/08 C07D413/06 C07D417/06 C07D471/04 C07D307/81 A61K31/404 A61K31/4178 A61P25/00 A61P9/00 A61P1/00

Abstract RU 2459806 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to new substituted heteroaryl derivatives of general formula I: , wherein: A means N, CR^7-10, with A at the most twice meaning N; W means O, S or NR⁴, the values B, C, R^7-10 are presented in clause 1 of the patent claim. The method for preparing the compound I is described.

EFFECT: compounds show analgesic activity that enables using them for a variety of diseases, especially acute pain, neuropathic, chronic or inflammatory pain.

16 cl, 2 tbl, 307 ex

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RU 2 459 806 C2

Authors

Tsemol'Ka Zaskja

Shunk Shtefan

Ehngl'Berger Verner

Kegel' Babette-Ivonne

Lints Klaus

Shik Khans

Zonnenshajn Khel'Mut

Graubaum Khajnts

Khintse Klaudia

Dates

2012-08-27—Published

2007-07-17—Filed