N1/N2-LACTAM ACETYL-CoA-CARBOXYLASE INHIBITORS Russian patent published in 2015 - IPC C07D471/20 C07D519/00 A61K31/438 A61K31/4709 A61K31/4725 A61P1/16 A61P3/10 

Abstract RU 2540337 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a compound of formula or its pharmaceutically acceptable salt, wherein G represents a group of formula or R1 represents isopropyl or tert-butyl; R2 represents naphthyl, quinolinyl or isoquinolinyl, R2 is optionally independently substituted by one-two groups of methyl, methoxy or chloro; R3 represents hydrogen. The invention also refers to a pharmaceutical composition containing the compound of formula (I).

EFFECT: compounds of formula (I) as acetyl-CoA-carboxylase(s) inhibitors.

6 cl, 10 dwg, 7 tbl, 125 ex

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RU 2 540 337 C2

Authors

Bagley Scott William

Dow Robert Lee

Griffith David Andrew

Smith Aaron Christopher

Dates

2015-02-10Published

2011-10-18Filed