FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to a compound of formula or its pharmaceutically acceptable salt, wherein G represents a group of formula or R1 represents isopropyl or tert-butyl; R2 represents naphthyl, quinolinyl or isoquinolinyl, R2 is optionally independently substituted by one-two groups of methyl, methoxy or chloro; R3 represents hydrogen. The invention also refers to a pharmaceutical composition containing the compound of formula (I).
EFFECT: compounds of formula (I) as acetyl-CoA-carboxylase(s) inhibitors.
6 cl, 10 dwg, 7 tbl, 125 ex
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Authors
Dates
2015-02-10—Published
2011-10-18—Filed