CONTRAST AGENT FOR INTRODUCTION OF FLUORINE-19 LABEL INTO PROTEINS CONTAINING LYSINE RESIDUES Russian patent published in 2016 - IPC A61K49/06 C07D333/36 

Abstract RU 2599500 C1

FIELD: medicine; pharmacology.

SUBSTANCE: invention relates to pharmacology and medical diagnostics. Disclosed is a contrast agent, representing N-(2,3,5-trifluoro-4,6-bis(trifluoromethyl)phenyl)-homocysteine thiolactone, which can be used for introduction of fluorine-19 label into protein molecules containing lysine residues.

EFFECT: invention provides higher quality and stability of a contrast agent.

1 cl, 1 dwg, 3 ex

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RU 2 599 500 C1

Authors

Godovikova Tatyana Sergeevna

Silnikov Vladimir Nikolaevich

Platonov Vyacheslav Evdokimovich

Chubarov Aleksej Sergeevich

Dates

2016-10-10Published

2015-08-04Filed