NEW AND EFFECTIVE DOSAGE FORMS OF TAPENTADOL Russian patent published in 2016 - IPC A61K31/137 A61K31/485 A61K45/06 A61P29/00 A61P25/04 

Abstract RU 2599846 C2

FIELD: medicine.

SUBSTANCE: present invention provides a combination for treating pain containing tapentadol and at least one opioid antagonist that includes naloxone or naltrexone (6 variants); a method of treating pain using the said combination (2 variants), a kit for treating pain that contains tapentadol and at least one opioid antagonist that includes naloxone or naltrexone.

EFFECT: higher efficiency and/or reduced side effects of tapentadol (for example, nausea and vomiting).

31 cl, 17 dwg

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RU 2 599 846 C2

Authors

Ramesh Sesha

Dates

2016-10-20Published

2009-10-29Filed