INHIBITORS OF PHOSPHODIESTERASE 10 ENZYME Russian patent published in 2018 - IPC C07D487/04 A61K31/4985 A61K31/502 A61P25/00 

Abstract RU 2667058 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel derivatives of formula (I), also to pharmaceutical compositions containing such compounds, to methods for preparing such compounds and compositions, to the use of such compounds or pharmaceutical compositions for the prevention or treatment of neurological, psychiatric and metabolic disorders and diseases. (I).

EFFECT: technical result: obtaining novel compounds which are inhibitors of the phosphodiesterase 10 (PDE10) enzyme and which may be useful for the treatment or prevention of neurological, psychiatric and metabolic disorders involving the PDE10 enzyme.

13 cl, 8 tbl

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RU 2 667 058 C2

Authors

Leklerk Loran Kristian L.

Bartolome-Nebreda Khose Manuel

Konde-Sejde Susana

Van Gol Mikhil Lyuk Mariya

Dates

2018-09-14Published

2013-07-08Filed