IMIDAZOLYL PROGESTERONE ANTAGONISTS Russian patent published in 2019 - IPC C07J43/00 A61K31/58 A61P15/04 A61P35/00 

Abstract RU 2679445 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound having the structure of formula (I) in which X is O, R1 is a hydrogen atom; R2 represents a hydrogen atom; R3 is hydrogen atom; R4 is a hydrogen atom; R5 is an N-imidazolyl group; R6 is a hydroxyl group; R7 is a radical of formula CnFmHo, wherein n is 2, 3, 4, 5 or 6, wherein m ≥ 1 and m+o = 2n + 1. Invention also relates to a method for treating a subject using a progesterone antagonist.

.

EFFECT: technical result: novel compounds of formula (I), that exhibit progesterone antagonism are obtained.

3 cl, 2 dwg, 1 tbl, 2 ex

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RU 2 679 445 C2

Authors

Nikish Klaus

Elger Valter

Santamma Bindu

Dates

2019-02-11Published

2014-06-05Filed