FIELD: medicine; pharmaceuticals.
SUBSTANCE: invention relates to an eremomycin derivative which can be used in medicine and pharmaceutical industry, corresponding to formula:
,
where Py – independently denotes pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, n=1–3, as well as its quaternized N-C10-20alkyl derivatives, hydrates, pharmacologically acceptable salts.
EFFECT: novel derivatives of eremomycin effective for treating bacterial infections caused by gram-positive bacteria.
4 cl, 11 ex, 2 tbl
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Authors
Dates
2019-12-10—Published
2019-01-23—Filed