3-ISOPROPOXY-6-R-IMIDAZO[1,2-B][1,2,4,5]TETRAZINES HAVING ANTIBACTERIAL ACTIVITY AGAINST NEISSERIA GONORRHOEAE Russian patent published in 2022 - IPC C07D487/04 A61K31/395 A61P31/04 

Abstract RU 2767869 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel 3-isopropoxy-6-R-imidazo[1,2-b][1,2,4,5]tetrazines of general formula

where R = hydrogen (1a), benzylthio (1b).

EFFECT: novel compounds are obtained, which are active against gram-negative bacteria Neisseria gonorrhoeae.

1 cl

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RU 2 767 869 C1

Authors

Charushin Valerij Nikolaevich

Ignatenko Nina Konstantinovna

Ishmetova Rashida Irshotovna

Gerasimova Natalya Avenirovna

Evstigneeva Natalya Petrovna

Zilberberg Natalya Vladimirovna

Kungurov Nikolaj Vasilevich

Rusinov Gennadij Leonidovich

Chupakhin Oleg Nikolaevich

Dates

2022-03-22Published

2020-12-18Filed