INHIBITOR OF MATRIX METALLOPROTEINASES OF 2nd AND 9th TYPES FROM SERIES OF BENZOYLAMINO(PHENYLSULPHONYL)-L-OXYPROLINE DERIVATIVES, HAVING NEUROPROTECTIVE AND ANTICANCER ACTIVITY Russian patent published in 2024 - IPC C07D207/48 A61K31/401 A61P35/00 A61P25/00 

Abstract RU 2826902 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel compound 1-({4-[(2,4-dichlorobenzoyl)amino]phenyl}sulphonyl-(2S,4R)-4-hydroxypyrrolidine-2-carboxylic acid.

EFFECT: new compound 1-({4-[(2,4-dichlorobenzoyl)amino]phenyl}sulfonyl-(2S,4R)-4-hydroxypyrrolidine-2-carboxylic acid is obtained which has neuroprotective and anticancer activity.

1 cl, 8 dwg, 4 tbl, 5 ex

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RU 2 826 902 C1

Authors

Grigorkevich Oksana Sergeevna

Mokrov Grigorij Vladimirovich

Nikolaev Sergej Vladimirovich

Antipova Tatyana Alekseevna

Kovalenko Larisa Petrovna

Gudasheva Tatyana Aleksandrovna

Durnev Andrej Dmitrievich

Dorofeev Vladimir Lvovich

Dates

2024-09-18Published

2023-07-14Filed