20-AROYL-12-HYDROXY-17,17-DIMETHYL-3-PHENYL-3,10,13- TRIAZAPENTACYCLO-[10.7.1.0.0.0]-E ICOSA-4,6,8,14(19)-TETRAENE-2,11,15-TRIONES AND METHOD FOR THEIR PREPARING Russian patent published in 2005 - IPC

Abstract RU 2257386 C1

FIELD: organic chemistry, chemical technology.

SUBSTANCE: invention relates to new individual compounds of azapentacycloeicosanes class. Invention describes 20-aroyl-12-hydroxy-17,17-dimethyl-3-phenyl3,10,13-triazapentacyclo[10.7.1.01,10.O4,9.O14,19]eicosa-4,6,14(19)-2,11,15-triones of the formula:

wherein R means hydrogen atom; Ar means phenyl; or R means benzyl and Ar means p-methoxyphenyl group. Also, the invention describes a method for preparing these compounds. Invention provides preparing new compounds that can be used as the parent substances for synthesis of new heterocyclic systems.

EFFECT: improved preparing method, valuable chemical properties of compounds.

4 cl, 1 tbl, 3 ex

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RU 2 257 386 C1

Authors

Mashevskaja I.V.

Duvalov A.V.

Bozdyreva K.S.

Klinchina M.L.

Dyrenkov R.O.

Maslivets A.N.

Dates

2005-07-27Published

2004-05-05Filed