FIELD: organic chemistry, medicine, pharmacology, pharmacy.
SUBSTANCE: invention relates to an agent eliciting immunomodulating, antitumor, bacteriostatic and anti-aggregation properties and representing 1-hexadecyl-R-(-)-3-oxy-1-azoniabicyclo[2.2.2]octane bromide and a method for its synthesis. Method involves quartenization of R-(-)-azabicyclo[2.2.2]octane-3-ol with hexadecyl bromide at heating in organic solvent medium. Agent shows low toxicity, high effectiveness, it doesn't cause allergic effect and doesn't possess cumulative effect.
EFFECT: valuable medicinal properties of agent.
3 cl, 9 dwg, 6 tbl, 2 ex
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METHOD FOR PREPARING 1-HEXADECYL-R-(-)-3-HYDROXY-1-AZONIABICYCLO[2.2.2]OCTANE BROMIDE - IMMUNOMODULATOR ELICITING ANTITUMOR, BACTERIOSTATIC AND ANTI-AGGREGATIVE PROPERTIES | 2005 |
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Authors
Dates
2007-04-10—Published
2005-04-28—Filed