METHOD OF RACEMATION OF (S)-(+) AND (R)-(-)-10,11-DIHYDRO-10-HYDROXY-5H-DEBENZ(b,f)AZEPIN-5-CARBOXAMIDE AND THEIR OPTICALLY ENRICHED MIXTURES Russian patent published in 2009 - IPC C07D223/28 C07D223/22 A61K31/55 

Abstract RU 2345986 C2

FIELD: chemistry.

SUBSTANCE: present invention pertains to methods of obtaining compounds V and VI , methods of racemation of optically pure or optically enriched compounds I and II , intermediate product VII , used in the process of obtaining I and II compounds. The invention also relates to methods of making compounds with general formula VIII and IX .

EFFECT: method of obtaining and racemation of useful biologically active compounds distinguished by simple design, availability and cheapness of initial reagents and high output.

15 cl, 5 ex

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RU 2 345 986 C2

Authors

Lermont Dehvid Aleksander

Dates

2009-02-10Published

2004-05-11Filed