FIELD: chemistry.
SUBSTANCE: present invention pertains to methods of obtaining compounds V and VI , methods of racemation of optically pure or optically enriched compounds I and II , intermediate product VII , used in the process of obtaining I and II compounds. The invention also relates to methods of making compounds with general formula VIII and IX .
EFFECT: method of obtaining and racemation of useful biologically active compounds distinguished by simple design, availability and cheapness of initial reagents and high output.
15 cl, 5 ex
Title |
Year |
Author |
Number |
METHOD OF CONVERTING (S)-(+)-I (R)-(-)-10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/b,f/AZEPIN-5-CARBOXAMIDE AND OPTICALLY ENRICHED MIXTURES THEREOF |
2005 |
- Lermont Dehvid Aleksander
- Vajngertner Gjunter
- Kremer Mattias
|
RU2382772C2 |
METHODS FOR PREPARING OPTICALLY PURE (S)-(+)- AND/OR (R)-(-)-ISOMERS OF 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ[b,f]AZEPINE-5-CARBOXAMIDE, THEIR CORRESPONDING 10-ACETOXY-DERIVATIVES AND NOVEL INTERMEDIATE COMPOUNDS |
2002 |
- Lermont Dehvid Aleksander
|
RU2318813C2 |
ASYMMETRIC CATALYTIC REDUCTION OF OXCARBAZEPINE |
2006 |
- Lermont Dehvid Aleksander
- Grasa Gabr'Ela Aleksandra
- Tsanotti-Dzheroza Antonio
|
RU2439060C2 |
SUBSTITUTED DIHYDRODIBENZO[B,F]AZEPINES, METHOD OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION SHOWING ANTIEPILEPTIC ACTIVITY |
1996 |
- Zhan Benes
- Patrisio Manuehl V'Ejru Arauzho Suarish Da Silva
|
RU2168502C2 |
METHOD FOR PREPARING 10,11-DIHYDRO-1-HYDROXY-5H-DIBENZ[b,f]AXEPINE-5-CARBOXAMIDE AND 10,11-DIHYDRO-10-OXO-5H-DIBENZ[b,f]AZEPINE-5-CARBOXAMIDE |
2002 |
- Lermont Dehvid Aleksander
|
RU2311411C2 |
METHOD OF PRODUCING 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/b, f/AZEPINE-5-CARBOXAMIDE |
2006 |
- Lermont Dehvid Aleksander
- Vajngertner Gjunter
- Kremer Mattias
|
RU2418789C2 |
METHOD FOR PREPARING 10,11-DIHYDRO-10-OXO-5N-DIBENZ(b,f)AZEPINE-5-CARBOXAMIDE |
2007 |
- Lermont Dehvid Aleksander
|
RU2449992C2 |
NEW DERIVATIVES OF 10,11-DIHYDRO-10-OXO-5H-DIBENZO- -[B,F]AZEPINE-5- CARBOXAMIDE, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION, METHOD OF TREATMENT OF CONVULSANT STATES |
1997 |
- Benesh Jan
- Soares Da Silva Patrisio Manuehl V'Ejra Arauzho
- Learmont David Aleksandr
|
RU2187503C2 |
METHOD OF 5H-DIBENZ[B, FIAZEPINES SYNTHESIS |
1992 |
- Tokmakov Gennadij Petrovich
- Grandberg Igor' Iogannovich
|
RU2007395C1 |
METHODS FOR PRODUCTION OF RACEMIC AMINOSUBSTITUTED 5,6,7,8-TETRAHYDROQUINOLINE OR RACEMIC AMINOSUBSTITUTED 5,6,7,8-TETRAHYDROISOQUINOLINE, METHODS FOR SEPARATION AND RACEMIZATION THEREOF, METHODS FOR PRODUCTION OF KETOSUBSTITUTED 5,6,7,8-TETRAHYDROQUINOLINE OR KETOSUBSTITUTED 5,6,7,8-TETRAHYDROISOQUINOLINE, METHOD FOR PRODUCTION OF ENANTIOMER PF CONDENSED BYCYCLIC RING SUBSTITUTED WITH PRIMARY AMINE, 5,6,7,8-TETRAHYDROQUINOLINE DERIVATIVES |
2002 |
- Makichern Ehrnest Dzh.
- Bridzher Gari Dzh.
- Skupinska Kristina A.
- Skerldzh Renato T.
|
RU2308451C2 |