PHARMACEUTICAL COMPOSITION BASED ON 3-(4-METHYLIMIDAZOLE-1-YL)IMIDAZO[1,2-b][1,2,4,5]TETRAZINE AS ANTI-TUMOR AGENT Russian patent published in 2017 - IPC A61K31/395 A61K47/10 A61K47/16 

Abstract RU 2614234 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to pharmaceutical industry and includes pharmaceutical composition, which is solution of pharmaceutically acceptable substance 3-(4-methylimidazole-1-yl)imidazo[1,2-b][1,2,4,5]tetrazine of formula (I) and D-mannitol in water. Composition is used for therapy of malignant tumors in human or animal.

EFFECT: technical result is obtaining stable, long-term stored solution of Substance 1.

1 cl

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RU 2 614 234 C2

Authors

Danilenko Valerij Nikolaevich

Charushin Valerij Nikolaevich

Rusinov Gennadij Leonidovich

Markova Alina Aleksandrovna

Ishmetova Rashida Irshotovna

Abilev Serikbaj Karimovich

Ignatenko Nina Konstantinovna

Tolshchina Svetlana Gennadevna

Ratkin Anatolij Vasilevich

Shtil Aleksandr Albertovich

Dates

2017-03-23Published

2015-03-31Filed