FIELD: chemistry.
SUBSTANCE: invention relates to the field of organic chemistry, namely a cyclic amine derivative or a pharmacologically acceptable salt thereof of general formula (I), wherein the carbon atom marked with * is an asymmetric carbon atom and A is a group represented by the general formula (IIa), (IIb) or (IIc), where R1 is a methyl group or an ethyl group optionally substituted by a halogen atom, R2 represents a hydrogen atom or an alkylcarbonyl group having from 2 to 5 carbon atoms, each R3 independently represents a methyl group or an ethyl group, and n is 1 or 2. Invention also relates to a medicament, an analgesic and a therapeutic agent based on a compound of formula (I). , .
EFFECT: cyclic amine derivative having an analgesic effect is obtained, in particular with respect to neuropathic pain and/or fibromyalgia syndrome.
10 cl, 18 dwg, 8 tbl, 19 ex
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Authors
Dates
2018-09-14—Published
2016-02-26—Filed