METHOD FOR PREPARING 3-AROYLBENZO[d]PYRROLO[2,1-b]THIAZOL-1,2-DIONES EXHIBITING ANTIRADICAL ACTIVITY Russian patent published in 2023 - IPC C07D513/04 

Abstract RU 2806262 C1

FIELD: pharmacological products.

SUBSTANCE: invention is related to a method for producing 3-aroylbenzo[d]pyrrolo[2,1-b]thiazol-1,2-diones, which can be used as starting products for the synthesis of new heterocyclic systems and in pharmacology. The method involves the interaction of 3-aroylpyrrolo[2,1-c][1,4]benzothiazine-1,2,4-triones with diphenylcarbinol in an aprotic solvent (toluene) when heated at 113°C for 2 hours:

I, III: Ar = C6H5 (a); Ar = C6H4Me-4 (b); Ar = C6H4Cl-4 (c).

EFFECT: development of a simple method for synthesis of 3-aroylbenzo[d]pyrrolo[2,1-b]thiazole-1,2-diones.

1 cl, 1 tbl, 4 ex

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RU 2 806 262 C1

Authors

Maslivets Andrei Nikolaevich

Khramtsova Ekaterina Evgenevna

Lystsova Ekaterina Aleksandrovna

Dates

2023-10-30Published

2023-03-16Filed