Show metadata Hide metadata

(19)

(11)

2 613 633

(13)

(51)

IPC

C07D407/06(2006-01-01)

C07D413/06(2006-01-01)

A61K31/353(2006-01-01)

A61K31/5377(2006-01-01)

A61P31/06(2006-01-01)

(21) (22)

Application

2016108546, 2016-03-09

(24)

Start date

2016-03-09

(22)

Actual filing date

2016-03-09

(45)

Published

2017-03-21

(72)

Inventor

Chernov Nikita MaksimovichYakovlev Igor PavlovichShutov Roman VadimovichVinogradova Tatyana IvanovnaManicheva Olga AlekseevnaDogonadze Marine ZaurievnaZabolotnykh Nataliya VyacheslavovnaVitovskaya Mariya Lvovna

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennaya Khimiko-Farmatsevticheskaya Akademiya" Ministerstva Zdravookhraneniya Rossijskoj Federatsii Vo Spkhfa Minzdrava Rossii)

CHLORIDE 4-[(1E)-1-(6-CHLORO-4-OXO-4N-CHROMEN-3-YL)-4-METHYLPENT-1-EN-3-YL]MORPHOLINE-4-YL, METHOD OF PRODUCING THEREOF AND ITS ANTITUBERCULOSIS EFFECT Russian patent published in 2017 - IPC C07D407/06 C07D413/06 A61K31/353 A61K31/5377 A61P31/06

Abstract RU 2613633 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry, namely to chloride 4-[(1E)-1-(6-chloro-4-oxo-4H-chromen-3-yl)-4-methylpent-1-en-3-yl]morpholine-4-yl of formula I

and method of producing thereof.

EFFECT: new heterocyclic compound, may be used as a potential antituberculosis drug.

3 cl, 5 dwg, 2 tbl, 2 ex

Similar patents RU2613633C1

Title	Year	Author	Number
(4-(3-HYDROXYPHENYL)PIPERAZINE-1-YL)(5-NITROFURAN-2-YL)METHANON, WHICH HAS ANTITUBERCULAR ACTIVITY AGAINST THE CAUSATIVE AGENT OF MULTIDRUG-RESISTANT TUBERCULOSIS, AND THE METHOD FOR ITS PREPARATION	2021	Dobrikov Georgi Dogonadze Marine Zaurievna Soloveva Natalya Sergeevna Vyazovaya Anna Aleksandrovna Vlcheva Violeta Mokrousov Igor Vladislavovich Zhuravlev Vyacheslav Yurevich	RU2784399C1
SELECTIVE ANTI-TUBERCULOSIS AGENTS, REPRESENTING 3-AMINOSUBSTITUTED 6-(3,5-DIMETHYLPYRAZOL-1-YL)-1,2,4,5-TETRAZINES	2012	Rusinov Gennadij Leonidovich Fedorova Ol'Ga Vasil'Evna Ishmetova Rashida Irshotovna Ganebnykh Il'Ja Nikolaevich Ovchinnikova Irina Georgievna Kravchenko Marionella Anatol'Evna Charushin Valerij Nikolaevich	RU2519218C2
1-ETHYL-6-FLUORO-4-OXO-7-(8-ETHOXY-2-OXO-2H-CHROMEN-3-YL)-1,4-DIHYDROQUINOLINE-3-CARBOXYLIC ACID WITH ANTI-TUBERCULAR ACTIVITY	2017	Charushin Valerij Nikolaevich Mochulskaya Nataliya Nikolaevna Kotovskaya Svetlana Konstantinovna Kravchenko Marionella Anatolevna Skornyakov Sergej Nikolaevich Medvinskij Igor Davydovich	RU2642426C1
DIALKYL(2-METHYL-4-OXOPENT-2-YL)PHOSPHINE OXIDE PYRIDINOYL HYDRAZONES, HAVING ANTITUBERCULOUS ACTIVITY	2012	Kostin Anton Alekseevich Tatarinov Dmitrij Anatol'Evich Kashapov Lenar Ramilovich Chestnova Regina Valer'Evna Valiev Ravil' Shamilovich Garaev Ramil Sufiakhmetovich Buzykin Boris Ivanovich Mironov Vladimir Fedorovich	RU2498990C1
3-TRIAZENONE INDOLES POSSESSING MYCOBACTERIUM ACTIVITY	2016	Apt Aleksandr Solomonovich Velezheva Valeriya Sergeevna Nikonenko Boris Vladimirovich Kornienko Albert Grigorevich Majorov Konstantin Borisovich Ivanov Pavel Yurevich Kondrateva Tatyana Konstantinovna Korotetskaya Marina Valerevna Salina Elena Gennadevna	RU2724334C1
5-FLUORO-2-(4-ETHOXYCARBONYLDIPIPERAZINE-1-YL)-1,3-BENZOTHIAZINE-4-ONE, WHICH HAS ANTI-TUBERCULOSIS ACTIVITY	2018	Charushin Valerij Nikolaevich Nosova Emiliya Vladimirovna Poteeva Anna Dmitrievna Kotovskaya Svetlana Konstantinovna Lipunova Galina Nikolaevna Kravchenko Marionella Anatolevna Skornyakov Sergej Nikolaevich Medvinskij Igor Davydovich	RU2663848C1
SELECTIVE ANTITUBERCULOSIS AGENT REPRESENTING 3-HYDRAZONO-6-(3,5-DIMETHYLPYRAZOL-1-YL)- 1,2,4,5-TETRAZINE AND METHOD FOR PREPARING IT	2011	Rusinov Gennadij Leonidovich Fedorova Ol'Ga Vasil'Evna Ishmetova Rashida Irshotovna Ganebnykh Il'Ja Nikolaevich Ovchinnikova Irina Georgievna Kravchenko Marionella Anatol'Evna Charushin Valerij Nikolaevich	RU2479311C2
COMPOUND OF 8-(4-METHYL-4H-1,2,4-TRIAZOL-3-YL)-6-(METHYLSULPHONYL)-2-(5-NITRO-2-FUROYL)-2,6-DIAZASPIRO[3.4]OCTANE, HAVING ANTI-TUBERCULOSIS ACTIVITY AGAINST MULTIDRUG-RESISTANT TUBERCULOSIS AGENT, AND METHOD FOR PRODUCTION THEREOF	2023	Lukin Aleksej Yurevich Vinogradova Tatyana Ivanovna Dogonadze Marine Zaurievna Komarova Kristina Yurevna Vinogradova Lyubov Vladimirovna Darin Dmitrij Viktorovich Lavrova Anastasiya Igorevna Postnikov Evgenij Borisovich Sychev Aleksandr Vladimirovich Yablonskij Petr Kazimirovich	RU2825646C1
ANTITUBERCULOSIS AGENT BASED ON 4'-HYDROXY-1'-(2-HYDROXYPHENYL)-3'-ACYL-SPIRO[BENZO[b][1,4]THIAZINE-2,2'-PYRROLE]-3,5'(1 'H,4H)-DIONES	2023	Balandina Svetlana Iurevna Lukmanova Dzhamilia Nailevna Mashevskaia Irina Vladimirovna	RU2806097C1
DIMEPHOSPHONE ISONICOTINOYLHYDRAZONE WITH ANTI-TUBERCULOSIS ACTIVITY	2011	Buzykin Boris Ivanovich Nabiullin Vazikh Nurulaevich Mironov Vladimir Fedorovich Chestnova Regina Valer'Evna Garaev Ramil Sufiakhmetovich Kashapov Lenar Ramilovich Mironova Ekaterina Vladimirovna Tatarinov Dmitrij Anatol'Evich Kostin Anton Alekseevich	RU2457212C1

RU 2 613 633 C1

Authors

Chernov Nikita Maksimovich

Yakovlev Igor Pavlovich

Shutov Roman Vadimovich

Vinogradova Tatyana Ivanovna

Manicheva Olga Alekseevna

Dogonadze Marine Zaurievna

Zabolotnykh Nataliya Vyacheslavovna

Vitovskaya Mariya Lvovna

Dates

2017-03-21—Published

2016-03-09—Filed